13:40 - 15:10
Room: ANA Crowne Plaza “Ohtori” Room C
Workshop Session
Chair/s:
Cem Gabay, Hiroki Yoshida
Structure of an engineered IFN-λ/IFN-λR1/IL-10Rβ complex provides insight into the functional dichotomy of type III versus type I IFNs
Juan Luis Mendoza1, William M Schneider2, Hans-Heinrich Hoffman2, Koen Vercauteren2, Kevin M Jude1, Anming Xiong3, Ignacio Moraga1, Tim M Horton1, Jeffrey S Glenn3, Ype P de Jong2, 4, K Christopher Garcia1
1Howard Hughes Medical Institute, Department of Molecular and Cellular Physiology and Department of Structural Biology, Stanford University School of Medicine, Stanford, CA 94305, USA, Stanford, United States, 2Laboratory of Virology and Infectious Disease, The Rockefeller University, New York, NY 10065, USA, New York, United States, 3Department of Medicine, Division of Gastroenterology and Hepatology, Department of Microbiology and Immunology, Stanford University School of Medicine, Stanford, CA 94305, USA Stanford University School of Medicine, Stanford, CA 94305, USA, Stanford, United States, 4Center for the Study of Hepatitis C, Division of Gastroenterology and Hepatology, Weill Cornell Medicine, New York, NY 10065, USA, New York, United States

Type III interferons (IFN-λs) are cytokines that share a common signaling pathway, downstream target genes, antiviral and antiproliferative activities with type I IFNs, but drive these processes with less potency and via different cell surface receptors. The intrinsically low-affinity of IL-10Rβ, one of the two cognate IFN-λ receptors, was believed to be a limiting factor to crystallizing the wild-type signaling complex. Here, we report the crystal structure of the IFN-λ receptor ternary complex enabled by the in vitro evolution of a high-affinity IFN-λ to stabilize the complex. Structural and sequence analyses provide insights on the mechanism of IL-10Rβ engagement with IFN-λ and other IL-10 cytokines. We harnessed the enhanced affinity of our engineered IFN-λ as means to enhance the potency of STAT signaling, gene induction, and antiviral and antiproliferative activities. More importantly, an in vivo study of hepatitis B virus infected human-liver chimeric mice shows enhanced antiviral activity by our high-affinity IFN-λ without increased toxicity relative to the wild-type IFN-λ or untreated control mice. We provide evidence that IFN-λ antiviral activities can be improved through protein engineering, and suggest an avenue by which these promising molecules may be pursued for clinical use.


Reference:
Tu-WS11-5
Session:
Workshop 11, “Emerging cytokines”
Presenter/s:
Juan Luis Mendoza
Presentation type:
Oral Presentation
Room:
ANA Crowne Plaza “Ohtori” Room C
Chair/s:
Cem Gabay, Hiroki Yoshida
Date:
Tuesday, 31 October 2017
Time:
14:48 - 14:58
Session times:
13:40 - 15:10