17:00 - 19:00
Room: ANA Crowne Plaza “Ohtori” Room A
Evening Symposium
Chair/s:
Akinori Takaoka, Keiko Ozato
Chromatin binding factor BRD4 directs development of hematopoietic stem cells and regulates inflammatory responses in macrophages through super-enhancers
Keiko Ozato1, Wenjing Yang2, Ryoji Yagi3, Anne Gegonne4, Akira Nishiyama5, Jun Zhu2, Jingfang Zhu3, Dinah Singer4, Anup Dey1
1NICHD, NHLBI, 3 NIAID, 4NCI, National Institutes of Health 5. Yokohama City University, Bethesda, United States, 2NHLBI, National Institutes of Health, Bethesda, United States, 3NIAID,National Institutes of Health, Bethesda, United States, 4NCI, National Institutes of Health, Bethesda, United States, 5Yokohama City University, Yokohama, Japan

The bromodomain protein BRD4 binds to acetylated histones and. activates transcriptional elongation of many genes. BRD4 occupies the TSS, gene body and numerous enhancers, including super-enhancers. We investigated the role of BRD4 in the development and activity of innate immunity by testing conditional Brd4 knockout mice. Our work was promoted by a number of recent papers reporting that small molecule inhibitors for BRD4 inhibit BRD4-acetyl histone interaction, and suppress blood cancer growth and reduce inflammation. These drugs are, thus believed to offer new therapeutic avenues to complex diseases. We show that Vav-Cre mediated Brd4 deletion in early embryos blocks the generation and differentiation of hematopoietic stem cells (HSCs). As a result, all immune cells, i.e., lymphocytes and myeloid cells as well as red blood cells were markedly reduced in Brd4 KO embryos leading to death in utero at around day 17- day18. This and additional data with later Brd4 deletion indicate that BRD4 is required for proliferation of developing immune cells at various stages. Brd4 deletion in post-mitotic macrophages displayed a less dramatic phenotype: induction of inflammatory cytokines and chemokines by LPS was only partially affected in Brd4 KO macrophages. ChIP-Seq analyses showed that BRD4 clusters on super-enhancers located near the genes controlling the myeloid lineage and inflammatory responses. Together, BRD4 affects every step of immune cell development and exerts complex regulatory influences on inflammation.


Reference:
Mo-ES1-4
Session:
Evening Symposium “Cytokines/IFNs in infection” incorporation with Hokkaido University and JSICR
Presenter/s:
Keiko Ozato
Presentation type:
Invited Speaker
Room:
ANA Crowne Plaza “Ohtori” Room A
Chair/s:
Akinori Takaoka, Keiko Ozato
Date:
Monday, 30 October 2017
Time:
18:12 - 18:36
Session times:
17:00 - 19:00